Sigma-LIGAND-1 (hydrochloride)
Sigma-LIGAND-1 hydrochloride is a selective sigma receptor ligand with an IC50s of 16 nM, 19 nM at the DTG site and the PPP site, respectively. Sigma-LIGAND-1 hydrochloride has a Ki of 4000 nM at the dopamine D2 receptor[1].
Product Specifications
CAS Number
[139652-86-1]
UNSPSC
12352005
Target
Sigma Receptor
Type
Reference compound
Related Pathways
Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/sigma-ligand-1-hydrochloride.html
Purity
99.13
Solubility
DMSO : 12.5 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
O=C1C(C)=C(C2=CC=CC=C2)OC3=CC=C(OCCCCCCN4CCC(O)CC4)C=C13.[H]Cl
Molecular Formula
C27H34ClNO4
Molecular Weight
472.02
References & Citations
[1]Erickson RH, et al. (Aminoalkoxy) chromones. Selective sigma receptor ligands. J Med Chem. 1992 May 1;35 (9) :1526-35.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Explore Other Products
Browse additional items from our catalog
![Mouse Monoclonal CD160 Antibody (688327) [DyLight 594]](https://cdn.genprice.uk/genprice/uk/genprice4.webp)
Mouse Monoclonal CD160 Antibody (688327) [DyLight 594]
![(7α,8β,9α,10α) -7,8,9,10-Tetrahydrobenzo[a]pyrene-7,8,9,10-tetrol-d8](https://cdn.genprice.uk/genprice/uk/genprice2.webp)
(7α,8β,9α,10α) -7,8,9,10-Tetrahydrobenzo[a]pyrene-7,8,9,10-tetrol-d8
Mouse Monoclonal HSP27 Antibody (8A7) [DyLight 755]
CHST5 (Carbohydrate sulfotransferase 5, Galactose/N-acetylglucosamine/N-acetylglucosamine 6-O-sulfotransferase 4-alpha, Intestinal N-acetylglucosamine-6-O-sulfotransferase, N-acetylglucosamine 6-O-sulfotransferase 3) (FITC)
TSPY1, CT (TSPY1, TSPY, Testis-specific Y-encoded protein 1, Cancer/testis antigen 78) (MaxLight 405) discontinued