GCPII-IN-1 (TFA)
GCPII-IN-1 (Compound 2) TFA is a GCPII (also known as PSMA) inhibitor scaffold with a Ki of 44.3 nM. GCPII-IN-1 TFA can be used in the research of prostate cancer[1].
Product Specifications
CAS Number
[1269794-89-9]
UNSPSC
12352211
Hazard Statement
H302, H315, H319
Target
Carboxypeptidase; PSMA
Type
Reference compound
Related Pathways
Immunology/Inflammation; Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gcpii-in-1-tfa.html
Purity
99.58
Solubility
H2O : 160 mg/mL (ultrasonic)
Smiles
OC(C(F)(F)F)=O.NCCCC[C@@H](C(O)=O)NC(N[C@H](C(O)=O)CCC(O)=O)=O
Molecular Formula
C14H22F3N3O9
Molecular Weight
433.33
Precautions
H302, H315, H319
References & Citations
[1]Jan Tykvart, et al. Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. Bioorg Med Chem. 2014 Aug 1;22 (15) :4099-108.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture and light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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