GCPII-IN-1 (TFA)
Product Specifications
UNSPSC Description
GCPII-IN-1 TFA is a glutamate carboxypeptidase II (GCPII, or PSMA) inhibitor scaffold with a Ki of 44.3 nM[1].
Target Antigen
Carboxypeptidase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gcpii-in-1-tfa.html
Solubility
H2O : 160 mg/mL (ultrasonic)
Smiles
OC(C(F)(F)F)=O.NCCCC[C@@H](C(O)=O)NC(N[C@H](C(O)=O)CCC(O)=O)=O
Molecular Weight
433.33
References & Citations
[1]Jan Tykvart, et al. Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. Bioorg Med Chem. 2014 Aug 1;22(15):4099-108.
Shipping Conditions
Room Temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-139840A/GCPII-IN-1-TFA-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-139840A/GCPII-IN-1-TFA-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
1269794-89-9
Available Sizes
Curated Selection
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