GCPII-IN-1 (TFA)
GCPII-IN-1 (Compound 2) TFA is a GCPII (also known as PSMA) inhibitor scaffold with a Ki of 44.3 nM. GCPII-IN-1 TFA can be used in the research of prostate cancer[1].
Product Specifications
CAS Number
[1269794-89-9]
UNSPSC
12352211
Hazard Statement
H302, H315, H319
Target
Carboxypeptidase; PSMA
Type
Reference compound
Related Pathways
Immunology/Inflammation; Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gcpii-in-1-tfa.html
Purity
99.58
Solubility
H2O : 160 mg/mL (ultrasonic)
Smiles
OC(C(F)(F)F)=O.NCCCC[C@@H](C(O)=O)NC(N[C@H](C(O)=O)CCC(O)=O)=O
Molecular Formula
C14H22F3N3O9
Molecular Weight
433.33
Precautions
H302, H315, H319
References & Citations
[1]Jan Tykvart, et al. Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. Bioorg Med Chem. 2014 Aug 1;22 (15) :4099-108.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture and light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS7074975 Inquire
Recombinant Rhizobium leguminosarum bv.viciae ATP synthase subunit a (atpB), partial
Sign In for Pricing
View Details 
RC200543L1V 200 µL
LDOC1 (NM_012317) Human Tagged ORF Clone Lentiviral Particle
Sign In for Pricing
View Details 
MBS9929014 Inquire
Duck Eukaryotic Translation Initiation Factor 3 Subunit B (EIF3B) ELISA Kit
Sign In for Pricing
View Details MBS1327594-01 0.02 mg (E-Coli)
Recombinant Bovine Multiple myeloma tumor-associated protein 2 homolog (MMTAG2)
Sign In for Pricing
View Details MBS1327594-02 0.1 mg (E-Coli)
Recombinant Bovine Multiple myeloma tumor-associated protein 2 homolog (MMTAG2)
Sign In for Pricing
View Details 
MBS1327594-03 0.02 mg (Yeast)
Recombinant Bovine Multiple myeloma tumor-associated protein 2 homolog (MMTAG2)
Sign In for Pricing
View Details