GPR132 antagonist 1

GPR132 antagonist 1 (GPR132-B-160, Compound 25) is a GPR132 antagonist with an EC50 value of 0.075 μM. GPR132 antagonist 1 has promote insulin secretion activity with an EC50 value of 0.7 μM[1].

Product Specifications

CAS Number

[898211-21-7]

UNSPSC

12352005

Target

G2A (GPR132)

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/gpr132-antagonist-1.html

Purity

99.72

Solubility

DMSO : ≥ 100 mg/mL

Smiles

O=C(C1=C(C)C2=C(C=CC(S(=O)(NCCC3=CC=CC=C3)=O)=C2)O1)O

Molecular Formula

C18H17NO5S

Molecular Weight

359.40

References & Citations

[1], . Gpcr. . CN116903563A.

Shipping Conditions

Blue Ice

Storage Conditions

-20°C, 3 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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