GPR132 antagonist 1
Product Specifications
UNSPSC Description
GPR132 antagonist 1 (GPR132-B-160, Compound 25) is a GPR132 antagonist with an EC50 value of 0.075 μM. GPR132 antagonist 1 has promote insulin secretion activity with an EC50 value of 0.7 μM[1].
Target Antigen
G2A (GPR132)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/gpr132-antagonist-1.html
Solubility
DMSO : ≥ 100 mg/mL
Smiles
O=C(C1=C(C)C2=C(C=CC(S(=O)(NCCC3=CC=CC=C3)=O)=C2)O1)O
Molecular Weight
359.40
References & Citations
[1]焦宁, 等. Gpcr调节剂及其应用. 专利. CN116903563A.
Shipping Conditions
Blue Ice
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-157189/GPR132-antagonist-1-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-157189/GPR132-antagonist-1-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
898211-21-7
Available Sizes
Curated Selection
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