GPR132 antagonist 1
GPR132 antagonist 1 (GPR132-B-160, Compound 25) is a GPR132 antagonist with an EC50 value of 0.075 μM. GPR132 antagonist 1 has promote insulin secretion activity with an EC50 value of 0.7 μM[1].
Product Specifications
CAS Number
[898211-21-7]
UNSPSC
12352005
Target
G2A (GPR132)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/gpr132-antagonist-1.html
Purity
99.72
Solubility
DMSO : ≥ 100 mg/mL
Smiles
O=C(C1=C(C)C2=C(C=CC(S(=O)(NCCC3=CC=CC=C3)=O)=C2)O1)O
Molecular Formula
C18H17NO5S
Molecular Weight
359.40
References & Citations
[1], . Gpcr. . CN116903563A.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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