Tigolaner-d4
Tigolaner-d4 is deuterium labeled Tigolaner. Tigolaner (BAY-1272858) acts on γ-aminobutyric acid (GABA) and glutamate-gated chloride channels. Tigolaner has antiparasitic activity[1][2].
Product Specifications
UNSPSC
12352005
Target
Chloride Channel; GABA Receptor; Isotope-Labeled Compounds; Parasite
Type
Isotope-Labeled Compounds
Related Pathways
Anti-infection; Membrane Transporter/Ion Channel; Neuronal Signaling; Others
Applications
COVID-19-immunoregulation
Field of Research
Infection; Neurological Disease
Solubility
10 mM in DMSO
Smiles
O=C(NC1(C#N)C([2H])([2H])C1([2H])[2H])C2=CC(C3=CN(C4=C(C(F)(F)F)C(C(F)(F)C(F)(F)F)=NN4C)N=C3)=CC=C2Cl
Molecular Formula
C21H9D4ClF8N6O
Molecular Weight
556.83
References & Citations
[1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216.|[2]The use ofstems in the selectionofInternationa Nonproprietary Names (INN) forpharmaceutical substances 2018 (Stem Book2018) .
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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