CP-866,087
CP-866,087 is a novel, potent and selective μ-opioid receptor antagonist with activity to inhibit opioid effects. CP-866,087 has shown promising preclinical efficacy data in disease models associated with alcohol consumption. CP-866,087 has also been used to study female sexual dysfunction[1].
Product Specifications
CAS Number
[519052-02-9]
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cp-866-087.html
Smiles
CC[C@@]1(C2=CC(NS(C)(=O)=O)=CC=C2)[C@]3([H])[C@@]1([H])CN(C3)CC4(CC5=CC=CC=C5C4)O
Molecular Formula
C24H30N2O3S
Molecular Weight
426.57
References & Citations
[1]Discovery of CP-866,087, a mu opioid receptor antagonist for the treatment of alcohol abuse and dependence
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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