CP-866,087
CP-866,087 is a novel, potent and selective μ-opioid receptor antagonist with activity to inhibit opioid effects. CP-866,087 has shown promising preclinical efficacy data in disease models associated with alcohol consumption. CP-866,087 has also been used to study female sexual dysfunction[1].
Product Specifications
CAS Number
[519052-02-9]
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cp-866-087.html
Smiles
CC[C@@]1(C2=CC(NS(C)(=O)=O)=CC=C2)[C@]3([H])[C@@]1([H])CN(C3)CC4(CC5=CC=CC=C5C4)O
Molecular Formula
C24H30N2O3S
Molecular Weight
426.57
References & Citations
[1]Discovery of CP-866,087, a mu opioid receptor antagonist for the treatment of alcohol abuse and dependence
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
Bovine Electron Transfer Flavoprotein Alpha Polypeptide ELISA Kit
![GABA A Receptor alpha 5 (GABRA5) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI1G5]](https://cdn.genprice.uk/products/937/68dd1b7d061270361ea1d1e6/imageurl/ta806598am.webp)