HENT4-IN-1
HENT4-IN-1 is a potent and selective human ENT4 (equilibrative nucleoside transporter 4) inhibitor with an IC50 of 74.4 nM[1].
Product Specifications
CAS Number
949467-71-4
UNSPSC
12352005
Target
Nucleoside Transporters
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/hent4-in-1.html
Concentration
10mM
Purity
99.94
Solubility
DMSO : ≥ 125 mg/mL
Smiles
CC(C)CN(C1=NC(NCCO)=NC2=C1N=C(NCCO)N=C2N(CC(C)C)CC(C)C)CC(C)C
Molecular Formula
C26H48N8O2
Molecular Weight
504.71
References & Citations
[1]Wang C, et al. Dipyridamole analogs as pharmacological inhibitors of equilibrative nucleoside transporters. Identification of novel potent and selective inhibitors of the adenosine transporter function of human equilibrative nucleoside transporter 4 (hENT4) . Biochem Pharmacol. 2013 Dec 1;86 (11) :1531-40.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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