Pentiapine
Pentiapine (CGS 10746) is a dopamine release inhibitor without binding to synaptic dopamine receptor sites[1][2].
Product Specifications
CAS Number
81382-51-6
Product Name Alternative
CGS 10746
UNSPSC
12352005
Target
Dopamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Pentiapine.html
Purity
99.95
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
CN1CCN(C2=NC3=CC=CC=C3SC4=NC=CN42)CC1
Molecular Formula
C15H17N5S
Molecular Weight
299.39
References & Citations
[1]Manzanedo C, et al. Effects of CGS 10746B on hyperactivity and place preference induced by morphine. Behav Brain Res. 2001 Nov 29;126 (1-2) :23-32.|[2]Bilsky EJ, et al. CGS 10746B, a novel dopamine release inhibitor, blocks the establishment of cocaine and MDMA conditioned place preferences. Pharmacol Biochem Behav. 1998 Jan;59 (1) :215-20.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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