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Protein kinase inhibitor 1 (hydrochloride)

Product Specifications

UNSPSC Description

Protein kinase inhibitor 1 hydrochloride is a potent HIPK2 inhibitor, with IC50s of 136 and 74 nM for HIPK1 and HIPK2, and a Kd of 9.5 nM for HIPK2.

Target Antigen

DYRK

Type

Reference compound

Related Pathways

Protein Tyrosine Kinase/RTK

Applications

Cancer-Kinase/protease

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/protein-kinase-inhibitor-1-hydrochloride.html

Purity

98.0

Solubility

DMSO : 8.33 mg/mL (ultrasonic)|H2O : 9.09 mg/mL (ultrasonic)

Smiles

O=C(NC/1=O)SC1=C\C2=CNC(C(C3=CC=C(N4CCNCC4)N=C3)=C2)=O.[H]Cl

Molecular Weight

419.89

References & Citations

[1]Miduturu CV, et al. High-throughput kinase profiling: a more efficient approach toward the discovery of new kinaseinhibitors. Chem Biol. 2011 Jul 29;18(7):868-79.EBioMedicine. 2021 Nov 24;74:103713.|EBioMedicine. 2022 Sep 28;85:104274.|J Biochem Mol Toxicol. 2021 Mar 9.

Shipping Conditions

Room Temperature

Storage Conditions

4°C (Powder, sealed storage, away from moisture)

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-U00439A/Protein-kinase-inhibitor-1-hydrochloride-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-U00439A/Protein-kinase-inhibitor-1-hydrochloride-SDS-MedChemExpress.pdf

Clinical Information

No Development Reported

CAS Number

2321337-71-5

Available Sizes

Curated Selection

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