PKR1 antagonist 1
PKR1 antagonist 1 (PC1) is a potent PKR1 antagonist. PKR1 antagonist 1 reduces hyperalgesia and allodynia in SNI mice[1].
Product Specifications
CAS Number
910113-60-9
UNSPSC
12352005
Target
Prokineticin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/pkr1-antagonist-1.html
Smiles
O=C1N=C(N(CC2=CC=C(C=C2)OC)C(N1CC3=CC=C(CC)C=C3)=O)NCCNC(N)=N
Molecular Formula
C23H29N7O3
Molecular Weight
451.52
References & Citations
[1]Guida F, et al. PC1, a non-peptide PKR1-preferring antagonist, reduces pain behavior and spinal neuronal sensitization in neuropathic mice. Pharmacol Res. 2015 Jan;91:36-46.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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