BCTP
BCTP is a TRPV1 antagonist. BCTP activated at low pH showed functional antagonist activity against human TRPV1 in CHO cells (IC50=18 nM) . BCTP can be used in the study of chronic pain[1].
Product Specifications
CAS Number
[464152-46-3]
UNSPSC
12352005
Target
TRP Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/bctp.html
Smiles
O=C(C1=CC(C2=CC=C(C=C2)Cl)=C(N=C1N3)C(C)(C)C)NC3=S
Molecular Formula
C17H16ClN3OS
Molecular Weight
345.85
References & Citations
[1]Culshaw A J, et al. Identification and biological characterization of 6-aryl-7-isopropylquinazolinones as novel TRPV1 antagonists that are effective in models of chronic pain[J]. Journal of medicinal chemistry, 2006, 49 (2) : 471-474.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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