PIKfyve-IN-1
PIKfyve-IN-1 is a highly potent and cell-active chemical probe that inhibits phosphatidylinositol-3phosphate 5-kinase (PIKfyve) with IC50 value of 6.9 nM. PIKfyve-IN-1 can be used for the research of PIKfyve in virology[1]. PIKfyve-IN-1 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
Product Specifications
CAS Number
[2857982-26-2]
UNSPSC
12352005
Hazard Statement
H302, H315, H318, H335
Target
PIKfyve
Type
Reference compound
Related Pathways
PI3K/Akt/mTOR
Applications
COVID-19-anti-virus
Field of Research
Cancer; Infection
Assay Protocol
https://www.medchemexpress.com/pikfyve-in-1.html
Purity
99.64
Solubility
DMSO : 100 mg/mL (ultrasonic; warming; heat to 80°C)
Smiles
NC1=NC=C(CCC2)C(C3=C2NC4=C3C=C(C#CCN(C)C)C=C4)=N1
Molecular Formula
C20H21N5
Molecular Weight
331.41
Precautions
H302, H315, H318, H335
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Explore Other Products
Browse additional items from our catalog
Capns2 sgRNA CRISPR Lentivector (Mouse) (Target 1)
CD79a (CD 79a, CD79A Antigen Immunoglobulin Associated alpha, CD79a Molecule Immunoglobulin Associated alpha, B Lymphocyte Specific MB1 Protein, B cell Antigen Receptor Complex Associated Protein alpha Chain, IGA, Ig alpha, Immunoglobulin Associated Alpha, Ly54, MB 1, MB 1 Membrane Glycoprotein, MB1, MB1 Membrane Glycoprotein, Membrane Bound Immunoglobulin Associated Protein, Surface IgM Associated Protein) (MaxLight 650)