Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

ML-030

ML-030 is a potent PDE4 inhibitor, with IC50 of 6.7 nM, 12.9 nM, 48.2 nM, 37.2 nM, 452 nM and 49.2 nM for PDE4A, PDE4A1, PDE4B1, PDE4B2, PDE4C1, and PDE4D2, respectively.

Product Specifications

CAS Number

1013750-77-0

UNSPSC

12352005

Target

Phosphodiesterase (PDE)

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/ML-030.html

Concentration

10mM

Purity

99.28

Solubility

DMSO : 50 mg/mL (ultrasonic)

Smiles

COC1=CC=C(C2=NN3C(SC2)=NN=C3C4=CC(OC)=CC=C4OC)C=C1OC

Molecular Formula

C20H20N4O4S

Molecular Weight

412.46

References & Citations

[1]Skoumbourdis AP, et al. Exploration and optimization of substituted triazolothiadiazines and triazolopyridazines as PDE4 inhibitors. Bioorg Med Chem Lett. 2009 Jul 1;19 (13) :3686-92.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

PDE4

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Automatic Tissue Processor BHTP-307
BHTP-307 1 Unit

Automatic Tissue Processor BHTP-307

Sign In for Pricing
View Details
Arsg Mouse Gene Knockout Kit (CRISPR)
KN501625 1 Kit

Arsg Mouse Gene Knockout Kit (CRISPR)

Sign In for Pricing
View Details
PITPNB Mouse Monoclonal Antibody [Clone ID: OTI6H10]
CF809305 100 µg

PITPNB Mouse Monoclonal Antibody [Clone ID: OTI6H10]

Sign In for Pricing
View Details
TRAP alpha (SSR1) Mouse Monoclonal Antibody (HRP conjugated) [Clone ID: OTI 4C9]
TA503267BM 100 µL

TRAP alpha (SSR1) Mouse Monoclonal Antibody (HRP conjugated) [Clone ID: OTI 4C9]

Sign In for Pricing
View Details
EXOSC1 Mouse Monoclonal Antibody [Clone ID: OTI1H9]
CF808518 100 µg

EXOSC1 Mouse Monoclonal Antibody [Clone ID: OTI1H9]

Sign In for Pricing
View Details
PE/Cyanine5 Anti-Human CD62L Antibody[HI62L]
E-AB-F1336G-01 20 Tests

PE/Cyanine5 Anti-Human CD62L Antibody[HI62L]

Sign In for Pricing
View Details