Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

A-887826

A-887826 is a potent, selective, oral bioavailable and voltage-dependent Na (v) 1.8 sodium channel blocker with an IC50 of 11 nM . A-887826 attenuates neuropathic tactile allodynia in vivo[1].

Product Specifications

CAS Number

1266212-81-0

UNSPSC

12352005

Hazard Statement

H301

Target

Sodium Channel

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/a-887826.html

Concentration

10mM

Purity

99.10

Solubility

DMSO : 250 mg/mL (ultrasonic)

Smiles

O=C(C1=CC(C2=CC=C(OCCCC)C(Cl)=C2)=CN=C1)NCC3=CC=CN=C3N4CCOCC4

Molecular Formula

C26H29ClN4O3

Molecular Weight

480.99

Precautions

H301

References & Citations

[1]Zhang XF, et al. A-887826 is a structurally novel, potent and voltage-dependent Na (v) 1.8 sodium channel blocker that attenuates neuropathic tactile allodynia in rats. Neuropharmacology. 2010 Sep;59 (3) :201-7.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

Nav1.8

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

basic Cytokeratin Mouse Monoclonal Antibody [Clone ID: SPM116]
AM33272PU-S 100 µg

basic Cytokeratin Mouse Monoclonal Antibody [Clone ID: SPM116]

Sign In for Pricing
View Details
Human TNNI3/cTn-I Antibody Pair Set
E-KAB-0128 50 µL & 100 µg

Human TNNI3/cTn-I Antibody Pair Set

Sign In for Pricing
View Details
XAB1 (GPN1) (NM_001145047) Human Over-expression Lysate
LC428661 20 µg

XAB1 (GPN1) (NM_001145047) Human Over-expression Lysate

Sign In for Pricing
View Details
C10orf63 (ENKUR) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI6F9]
TA804172AM 100 µL

C10orf63 (ENKUR) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI6F9]

Sign In for Pricing
View Details
Human TNFAIP8L3 activation kit by CRISPRa
GA117930 1 Kit

Human TNFAIP8L3 activation kit by CRISPRa

Sign In for Pricing
View Details
PTP rho (PTPRT) Human Gene Knockout Kit (CRISPR)
KN213847BN 1 Kit

PTP rho (PTPRT) Human Gene Knockout Kit (CRISPR)

Sign In for Pricing
View Details