(2R,3R) -GSK973
(2R,3R) -GSK973 is an isomer of GSK973. GSK973 is a highly selective, orally bioavailable inhibitor of the BD2s (second bromodomains) of the BET family[1].
Product Specifications
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/2r-3r-gsk973.html
Purity
99.91
Smiles
[H][C@]1([C@@H]2NC(C3=CC(C(NC)=O)=C4C([C@H]([C@@H](O4)CF)C5=CC=CC=C5)=C3)=O)[C@]2([H])COC1
Molecular Formula
C23H23FN2O4
Molecular Weight
410.44
References & Citations
[1]Preston A, et al. GSK973 Is an Inhibitor of the Second Bromodomains (BD2s) of the Bromodomain and Extra-Terminal (BET) Family. ACS Med Chem Lett. 2020;11 (8) :1581-1587. Published 2020 Jul 6.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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