AKR1C3-IN-1
AKR1C3-IN-1 is a potent, highly selective inhibitor of AKR1C3, with an IC50 of 13 nM.
Product Specifications
CAS Number
327092-81-9
UNSPSC
12352005
Hazard Statement
H315, H319, H335
Target
17β-HSD
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/AKR1C3-IN-1.html
Purity
98.21
Solubility
DMSO : ≥ 100 mg/mL
Smiles
O=S(N1CC2=CC=CC=C2CC1)(C3=CC(C(O)=O)=CC=C3)=O
Molecular Formula
C16H15NO4S
Molecular Weight
317.36
Precautions
H315, H319, H335
References & Citations
[1]Jamieson SM, et al. 3- (3,4-Dihydroisoquinolin-2 (1H) -ylsulfonyl) benzoic Acids: highly potent and selective inhibitors of the type 5 17-β-hydroxysteroid dehydrogenase AKR1C3. J Med Chem. 2012 Sep 13;55 (17) :7746-58.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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