A3AR antagonist 5
A3AR antagonist 5 (Compound 16) is a selective antagonist for human adenosine A3 receptor with an affinity pC of 4.542 μM[1].
Product Specifications
CAS Number
333436-43-4
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/a3ar-antagonist-5.html
Purity
98.17
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
O=C(CC1=CC=CC=C1)NC2=NC(C3=CC=C(OC)C=C3)=CS2
Molecular Formula
C18H16N2O2S
Molecular Weight
324.40
References & Citations
[1]Bhattacharya P, et al., Exploring 3D-QSAR of thiazole and thiadiazole derivatives as potent and selective human adenosine A3 receptor antagonists+. J Mol Model. 2005 Nov;11 (6) :516-24.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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