SI-2 (hydrochloride)
SI-2 (EPH 116 hydrochloride) is a highly promising SRC-3 inhibitor (PPI) . SI-2 (EPH 116 hydrochloride) has a much improved toxicity and pharmacokinetic profile, with acceptable oral availability[1].
Product Specifications
CAS Number
[1992052-49-9]
Product Name Alternative
EPH 116 (hydrochloride)
UNSPSC
12352005
Hazard Statement
H302, H315, H319
Target
Estrogen Receptor/ERR
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/si-2-hydrochloride.html
Purity
98.06
Solubility
DMSO : 5 mg/mL (ultrasonic)
Smiles
CN1C(N/N=C(C)/C2=CC=CC=N2)=NC3=CC=CC=C13.Cl
Molecular Formula
C15H16ClN5
Molecular Weight
301.77
Precautions
H302, H315, H319
References & Citations
[1]Song X, et al. Development of potent small-molecule inhibitors to drug the undruggable steroid receptor coactivator-3. Proc Natl Acad Sci U S A. 2016 May 3;113 (18) :4970-5.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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