CBP/p300-IN-12

Epigenetic Reader Domain; Histone Acetyltransferase

Reference compound

Epigenetics

Cancer

https://www.medchemexpress.com/cbp-p300-in-12.html

99.70

DMSO : 250 mg/mL (ultrasonic)

C=CC(NC1=CC=CC(NC(NC2=CC3=C([C@]4(OC(N(CC(N(CC5=CC=C(F)C=C5)[C@@H](C)C(F)(F)F)=O)C4=O)=O)CC3)C=C2)=O)=C1)=O

667.61

[1]Anthony Mastracchio, et al. Discovery of a Potent and Selective Covalent p300/CBP Inhibitor. ACS Med Chem Lett. 2021 Apr 5;12(5):726-731.

Room Temperature

-20°C, 3 years; 4°C, 2 years (Powder)

http://file.medchemexpress.com/batch_PDF/HY-132197/CBP-p300-IN-12-DataSheet-MedChemExpress.pdf

http://file.medchemexpress.com/batch_PDF/HY-132197/CBP-p300-IN-12-SDS-MedChemExpress.pdf

No Development Reported

2738688-57-6