CCG-63802
CCG-63802 is a selective, reversible and allosteric RGS4 inhibitor. CCG-63802 specifically binds to RGS4 and blocks the RGS4-Gαo interaction, with an IC50 value of 1.9 μM[1].
Product Specifications
CAS Number
[620112-78-9]
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
RGS Protein
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Cancer-programmed cell death
Field of Research
Cancer; Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/ccg-63802.html
Purity
98.83
Solubility
DMSO : 1.67 mg/mL (ultrasonic; warming)
Smiles
N#C/C(C1=NC2=CC=CC=C2S1)=C\C3=C(N=C4C(C)=CC=CN4C3=O)OC5=CC=CC(C)=C5
Molecular Formula
C26H18N4O2S
Molecular Weight
450.51
Precautions
H302, H315, H319, H335
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-70074/CCG-63802-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-70074/CCG-63802-SDS-MedChemExpress.pdf
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
RGS4
Available Sizes
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
