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ETP-46321

Product Specifications

CAS Number

1252594-99-2

Target

PI3K

Related Pathways

PI3K/Akt/mTOR signaling

Purity

0.998

Bioactivity

ETP-46321 is an effective and orally bioavailable PI3Kα/PI3Kδ inhibitor (Ki: 2.3/14.2 nM) .

Smiles

CS(=O)(=O)N1CCN(Cc2cn3cc(nc(N4CCOCC4)c3n2)-c2cnc(N)nc2)CC1

Molecular Formula

C20H27N9O3S

Molecular Weight

473.55

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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