LY2857785
Product Specifications
CAS Number
1619903-54-6
Target
Apoptosis, CDK
Related Pathways
Apoptosis, Cell Cycle/Checkpoint
Purity
0.9968
Bioactivity
LY2857785 is a type I competitive and reversible ATP kinase inhibitor against CDK7/CDK8/CDK9 (IC50s: 246 nM/16 nM/11 nM) .
Smiles
CC(C)c1n(C)nc2ccc(cc12)-c1ccnc(N[C@H]2CC[C@@H](CC2)NC2CCOCC2)n1
Molecular Formula
C26H36N6O
Molecular Weight
448.6
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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