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GNE-131

Product Specifications

CAS Number

1629063-81-5

Target

Sodium Channel

Related Pathways

Membrane transporter/Ion channel

Purity

0.9973

Bioactivity

GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM) .

Smiles

O=S(=O)(Nc1nnc2cc(OCC34CC5CC(CC(C5)C3)C4)c(cn12)C1CC1)C1CC1

Molecular Formula

C23H30N4O3S

Molecular Weight

442.57

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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