Stressin I
Product Specifications
Target
CRFR
Related Pathways
GPCR/G Protein
Bioactivity
Potent and selective corticotropin releasing factor receptor-1 (CRF1) agonist (Ki values are 1.5 and 224 nM for CRF1 and CRF2 receptors respectively) . Increases ACTH levels and increases faecal pellet output in vivo following i.p. administration.
Molecular Formula
C203H337N57O56
Molecular Weight
4472.24
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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