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Stressin I

Product Specifications

Target

CRFR

Related Pathways

GPCR/G Protein

Bioactivity

Potent and selective corticotropin releasing factor receptor-1 (CRF1) agonist (Ki values are 1.5 and 224 nM for CRF1 and CRF2 receptors respectively) . Increases ACTH levels and increases faecal pellet output in vivo following i.p. administration.

Molecular Formula

C203H337N57O56

Molecular Weight

4472.24

Shipping Conditions

Cool pack

Storage Temperature

-20°C

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