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SNX-482

Product Specifications

CAS Number

203460-30-4

Target

Calcium Channel

Related Pathways

Metabolism, Membrane transporter/Ion channel

Bioactivity

Potent and selective, voltage-dependent R-type CaV2.3 calcium channel blocker (IC50 = 30 nM) . Antinociceptive; inhibits nociceptive C-fibre and Aδ-fibre-evoked neuronal responses.

Molecular Formula

C192H274N52O60S7

Molecular Weight

4495.01

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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