Urantide acetate (669089-53-6 free base)
Product Specifications
CAS Number
9007-83-4
Target
Neurotensin Receptor
Related Pathways
GPCR/G Protein
Purity
0.9922
Bioactivity
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3) . Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors) .
Smiles
CC([C@@H](C(O)=O)NC([C@@H]1CSSC(C)([C@H](C(N[C@H](C(N[C@@H](C(N[C@H](C(N[C@H](C(N1)=O)Cc2ccc(O)cc2)=O)CCCN)=O)Cc(c[nH]3)c4c3cccc4)=O)Cc5ccccc5)=O)NC([C@H](CC(O)=O)N)=O)C)=O)C.CC(O)=O
Molecular Formula
C53H70N10O14S2
Molecular Weight
1135.31
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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