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Astressin 2B

Product Specifications

CAS Number

681260-70-8

Target

CFTR

Related Pathways

Membrane transporter/Ion channel

Bioactivity

Potent and selective corticotropin-releasing factor receptor 2 (CRF2) antagonist (IC50 values are 1.3 and > 500 nM for CRF2 and CRF1 respectively) . Antagonizes CRF2-mediated inhibition of gastric emptying.

Molecular Formula

C183H307N49O53

Molecular Weight

4041.69

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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