APETx2
Product Specifications
CAS Number
713544-47-9
Target
Sodium Channel
Related Pathways
Membrane transporter/Ion channel
Bioactivity
Acid-sensing ion channel 3 (ASIC3) channel blocker (IC50 values are 63 and 175 nM for homomeric rat and human ASIC3 channels) . Also inhibits NaV1.8 and NaV1.2 channels (IC50 values are 55 and 114 nM respectively) . Demonstrates analgesic properties against acid-induced and inflammatory pain.
Molecular Formula
C196H280N54O61S6
Molecular Weight
4561.06
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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