CTAP (TFA) (103429-32-9 free base)

CTAP (TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM. It displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somatostatin receptors. CTAP (TFA) (103429-32-9 free base) can be used for the study of L-DOPA-induced dyskinesia (LID)

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