M871

Selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM for GAL2 and GAL1 receptors respectively) . Blocks the pro-nociceptive effect of GAL2 receptor agonists.

C(=O)(N1[C@H](C(=O)N2[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N)=O)C)=O)CC(C)C)=O)C)=O)CC(C)C)=O)C)=O)CCC2)CCC1)[C@H]3N(C([C@H](CC4=CN=CN4)NC([C@@H](NC(=O)[C@H]5N(C(CNC([C@@H](NC([C@@H](NC([C@H](CC6=CC=C(O)C=C6)NC(CNC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CC=7C=8C(NC7)=CC=CC8)N)=O)[C@@H](C)O)=O)CC(C)C)=O)CC(N)=O)=O)CO)=O)C)=O)=O)=O)CC(C)C)=O)CC(C)C)=O)=O)CCC5)CCC(O)=O)=O)=O)CCC3