M1145

Product Specifications

CAS Number

1172089-00-7

Target

Neuropeptide Y Receptor

Related Pathways

Neuroscience|||GPCR/G Protein

Bioactivity

Potent and selective galanin receptor 2 (GAL2) agonist (EC50 = 38 nM, Ki values are 6.55, 497 and 587 nM at GAL2, GAL3 and GAL1 respectively) . Has an additive effect on the signal transduction of galanin.

Smiles

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