PL-017
Product Specifications
CAS Number
83397-56-2
Target
Opioid Receptor
Related Pathways
GPCR/G Protein, Neuroscience, Endocrinology/Hormones
Bioactivity
Selective μ opioid receptor agonist (IC50 values are 5.5 and > 10000 nM for inhibition of 125I-FK 33,824 and 125I-DADLE binding to μ and δ sites respectively) . Produces naloxone-reversible analgesia, catalepsy and hyperthermia following central administration in rats in vivo.
Smiles
C(N([C@H](C(=O)N1[C@@H](C(N)=O)CCC1)CC2=CC=CC=C2)C)(=O)[C@H]3N(C([C@H](CC4=CC=C(O)C=C4)N)=O)CCC3
Molecular Formula
C29H37N5O5
Molecular Weight
535.64
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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