RVD-Hp? acetate (1193362-76-3 free base)
Product Specifications
Target
Cannabinoid Receptor
Related Pathways
GPCR/G Protein
Purity
0.9987
Bioactivity
RVD-Hp? acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM) .
Smiles
CC(C)C[C@@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC1=CN=CN1)C(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H](C(C)C)NC(=O)[C@@H]3CCCN3C(=O)[C@H](CC(=O)O)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CCCN=C(N)N)N.CC(=O)O
Molecular Formula
C67H109N19O19
Molecular Weight
1484.71
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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