D[Leu4, Lys8]-VP acetate

D[Leu4, Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respectively. d[Leu4, Lys8]-VP acetate exhibits weak antidiuretic, vasopressor and oxytocic activiti

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