PKG inhibitor peptide
Product Specifications
CAS Number
82801-73-8
Target
PKA
Related Pathways
Tyrosine Kinase/Adaptors
Bioactivity
Competitive inhibitor of cGMP-dependent protein kinase (PKG) ; analog of a substrate peptide corresponding to a phosphorylation site of histone H2B. Competes with synthetic substrates (Ki = 86 mM) but does not inhibit phosphorylation of intact histones by PKG. Inhibits phosphorylation of intact histones by PKA.
Smiles
C[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CCCNC(N)=N)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(O)=O)C(O)=O
Molecular Formula
C38H74N18O10
Molecular Weight
943.12
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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