Kisspeptin 234 acetate (1145998-81-7 free base)
Product Specifications
Target
GPCR, Kisspeptin
Related Pathways
Endocrinology/Hormones, GPCR/G Protein
Purity
0.9934
Bioactivity
Kisspeptin 234 acetate (1145998-81-7 free base) is a Kisspeptin receptor (KISS1, GPR54) antagonist; a Kisspeptin-10 analogue. It inhibits the stimulation of inositol phosphate (IP) (IC50 = 7 nM) and the release of gonadotropin-releasing hormone (GnRH) by kisspeptin-10.
Smiles
C[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(NCC(N[C@@H](C(N[C@H](C(N[C@H](C(N)=O)CC1=CC=CC=C1)=O)CCCNC(N)=N)=O)CC2=CNC3=C2C=CC=C3)=O)=O)CC4=CC=CC=C4)=O)=O)CC(N)=O)=O)CC5=CNC6=C5C=CC=C6)=O)CC(N)=O)=O)NC(C)=O.CC(O)=O
Molecular Formula
C65H82N18O15
Molecular Weight
1355.46
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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