Dynorphin A (1-10)

Product Specifications

CAS Number

79994-24-4

Target

Opioid Receptor|||iGluR

Related Pathways

GPCR/G Protein|||Membrane transporter/Ion channel|||Neuroscience|||Endocrinology/Hormones

Bioactivity

Dynorphin A (1-10), an endogenous opioid neuropeptide, interacts with the ?-opioid receptor by binding to its extracellular loop 2 and inhibits NMDA-activated current, demonstrating an IC50 value of 42.0 ?M.

Smiles

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