C (Bua-Cpa-Thi-Val-Asn-Cys) -Pro-Agm

C (Bua-Cpa-Thi-Val-Asn-Cys) -Pro-Agm is a highly efficient, selective, and short-acting peptide V2 receptor agonist (V2R), with EC50s of hV2R and rV2R being 0.25 and 0.05 nM, respectively.

C(=O)(N1[C@H](C(N[C@@H](C(N(CC)CC)=O)CCCNC(=N)N)=O)CCC1)[C@H]2NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC3=CC=CS3)NC(=O)[C@H](CC4=CC=C(Cl)C=C4)NC(=O)CCCSC2