TAK-448

Product Specifications

CAS Number

1234319-68-6

Target

Kisspeptin

Related Pathways

GPCR/G Protein

Bioactivity

TAK-448 (MVT-602), a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM, has been studied in trials for the treatment of Prostate Cancer, Low Testosterone, Prostatic Neoplasms, and Hypogonadotropic Hypogonadism.

Smiles

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