UBP316
UBP316 (ACET) is a highly potent and selective kainate receptor GluK1 (GluR5) antagonist, with a Kb value of 1.4 nM. UBP316 is effective at blocking the depression of both field excitatory postsynaptic potentials (fEPSPs) and monosynaptically-evoked GABAergic transmission induced by ATPA, a GluK1 selective agonist[1].
Product Specifications
CAS Number
[936095-50-0]
Product Name Alternative
ACET
UNSPSC
12352005
Target
IGluR
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neurodegeneration
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ubp316.html
Purity
99.95
Solubility
1M NaOH : 80 mg/mL (ultrasonic; adjust pH to 11 with NaOH) |DMSO : 2 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
OC(C(SC(C1=CC=CC=C1)=C2)=C2CN3C(N(C=C(C)C3=O)C[C@H](N)C(O)=O)=O)=O
Molecular Formula
C20H19N3O6S
Molecular Weight
429.45
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
Lentiviral human WDSUB1 shRNA (UAS) - Lentiviral human WDSUB1 shRNA (UAS) (100)
Mouse Tumor Necrosis Factor alpha-Induced Protein 8-Like Protein 1 (TNFAIP8L1) ELISA Kit
Mouse Tumor Necrosis Factor alpha-Induced Protein 8-Like Protein 1 (TNFAIP8L1) ELISA Kit
Mouse Tumor Necrosis Factor alpha-Induced Protein 8-Like Protein 1 (TNFAIP8L1) ELISA Kit
