Opiranserin hydrochloride
Product Specifications
CAS Number
1440796-75-7
Target
GlyT, 5-HT Receptor, P2X Receptor
Related Pathways
Neuroscience, GPCR/G Protein, Membrane transporter/Ion channel
Purity
0.9933
Bioactivity
Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 μM) . It is development as an injectable agent for the treatment of postoperative pain.
Smiles
Cl.CCCCOc1c(OC)cc(cc1OC)C(=O)NCC1(CCOCC1)N(C)C
Molecular Formula
C21H35ClN2O5
Molecular Weight
430.97
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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