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TNIK-IN-5

Product Specifications

CAS Number

2754265-66-0

Target

Wnt/beta-catenin

Related Pathways

Cytoskeletal Signaling|||Stem Cells

Purity

0.9975

Bioactivity

TNIK-IN-5 is an potent TNIK inhibitor (IC50= 0.05 ?M) . TNIK-IN-5 potently inhibits Wnt signaling in intact cells. TNIK-IN-5 exhibits excellent in vitro anti-colorectal cancer activity.

Smiles

C(N1C=2C(=CC(=CC2)C=3C=C4C(=NC3)NC=C4)OC1=O)C5=CC(OC)=CC=C5

Molecular Formula

C22H17N3O3

Molecular Weight

371.39

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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