TNIK-IN-5
Product Specifications
CAS Number
2754265-66-0
Target
Wnt/beta-catenin
Related Pathways
Cytoskeletal Signaling|||Stem Cells
Purity
0.9975
Bioactivity
TNIK-IN-5 is an potent TNIK inhibitor (IC50= 0.05 ?M) . TNIK-IN-5 potently inhibits Wnt signaling in intact cells. TNIK-IN-5 exhibits excellent in vitro anti-colorectal cancer activity.
Smiles
C(N1C=2C(=CC(=CC2)C=3C=C4C(=NC3)NC=C4)OC1=O)C5=CC(OC)=CC=C5
Molecular Formula
C22H17N3O3
Molecular Weight
371.39
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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