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MRTX0902

Product Specifications

CAS Number

2654743-22-1

Target

Raf|||Ras

Related Pathways

GPCR/G Protein|||MAPK

Purity

0.9969

Bioactivity

MRTX0902 is an effective and high selective inhibitor of SOS1 with an IC50 of 46 nM and a Ki of 2 nM.

Smiles

C[C@@H](Nc1nnc(C)c2cnc(cc12)N1CCOCC1)c1cccc(C#N)c1C

Molecular Formula

C22H24N6O

Molecular Weight

388.47

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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