MRTX9768
Product Specifications
CAS Number
2629314-68-5
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9848
Bioactivity
MRTX-9768 is a synthetic lethal-based inhibitor designed to bind the PRMT5-MTA complex and selectively target MTAP/CDKN2A-deleted tumors.
Smiles
Cn1ncc(c1-c1c(F)cc2ccccc2c1C#N)-c1ccc2c(c1)c(CN)n[nH]c2=O
Molecular Formula
C24H17FN6O
Molecular Weight
424.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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