GSK3685032
Product Specifications
CAS Number
2170137-61-6
Target
DNA Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9949
Bioactivity
GSK3685032 is a non-covalent and selective DNMT1 inhibitor (IC50 = 36 nM) . The inhibitory effect is time-independent and reversible. GSK3685032 induces loss of DNA methylation and transcriptional activation and inhibits cancer cell growth.
Smiles
CCc1c(C#N)c(SC(C(N)=O)c2ccccc2)nc(N2CCC(N)CC2)c1C#N
Molecular Formula
C22H24N6OS
Molecular Weight
420.53
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS1406352-01 0.02 mg (E-Coli)
Recombinant Pseudoalteromonas haloplanktis Pyridoxine/pyridoxamine 5'-phosphate oxidase (pdxH)
Sign In for Pricing
View Details MBS1406352-02 0.1 mg (E-Coli)
Recombinant Pseudoalteromonas haloplanktis Pyridoxine/pyridoxamine 5'-phosphate oxidase (pdxH)
Sign In for Pricing
View Details MBS1406352-03 0.02 mg (Baculovirus)
Recombinant Pseudoalteromonas haloplanktis Pyridoxine/pyridoxamine 5'-phosphate oxidase (pdxH)
Sign In for Pricing
View Details MBS1406352-04 0.02 mg (Mammalian-Cell)
Recombinant Pseudoalteromonas haloplanktis Pyridoxine/pyridoxamine 5'-phosphate oxidase (pdxH)
Sign In for Pricing
View Details MBS1406352-05 1 mg (E-Coli)
Recombinant Pseudoalteromonas haloplanktis Pyridoxine/pyridoxamine 5'-phosphate oxidase (pdxH)
Sign In for Pricing
View Details MBS1406352-06 0.1 mg (Baculovirus)
Recombinant Pseudoalteromonas haloplanktis Pyridoxine/pyridoxamine 5'-phosphate oxidase (pdxH)
Sign In for Pricing
View Details