What is the catalog number for IRE1α kinase-IN-1?

The catalog number for IRE1α kinase-IN-1 is T9564.

What sizes are available for IRE1α kinase-IN-1?

IRE1α kinase-IN-1 is available in the following size(s): 1 mg, 5 mg, 1 mL - 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg.

How many pack sizes does IRE1α kinase-IN-1 come in?

IRE1α kinase-IN-1 is available in 7 different pack sizes.

Is IRE1α kinase-IN-1 in stock?

IRE1α kinase-IN-1 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures IRE1α kinase-IN-1?

IRE1α kinase-IN-1 is manufactured by Molfinity.

What is the estimated delivery time for IRE1α kinase-IN-1?

Estimated delivery time for IRE1α kinase-IN-1 is approximately 10 business day(s), depending on your location.

IRE1α kinase-IN-1

Product Specifications

CAS Number

2328097-41-0

Target

IRE1

Related Pathways

Cell Cycle/Checkpoint

Purity

0.997

Bioactivity

IRE1α kinase-IN-1 is a highly selective IRE1α (ERN1) inhibitor, with an IC50 of 77 nM, displaying 100-fold selectivity over the IRE1β isoform. It inhibits ER stress-induced IRE1α oligomerization and autophosphorylation, as well as IRE1α RNase activity (IC50=80 nM) .